Güncel Gönderiler: FEF, Kimya Bölümü Koleksiyonu
Toplam kayıt 455, listelenen: 61-80
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Determining the levels of acrylamide in some traditional foods unique to Turkey and risk assessment
(Brieflands, 2022)In this study, exposure risk assessment was made by determining the acrylamide levels of some traditional foods frequently consumed by the Turkish society and registered geographical indication. For this purpose, acrylamide ... -
Synthesis and in vitro α-glucosidase and cholinesterases inhibitory actions of water-soluble metallophthalocyanines bearing ({6-[3-(diethylamino)phenoxy]hexyl}oxy groups
(TUBITAK, 2022)In this paper, we have prepared peripherally tetra-({6-[3-(diethylamino)phenoxy]hexyl}oxy substituted cobalt(II), copper(II), manganese(III) phthalocyanines (3, 4, 5) and their water-soluble derivatives (3a, 4a, 5a). Then, ... -
Investigation of the usability of some triazole derivative compounds as drug active ingredients by ADME and molecular docking properties
(University Mohammed Premier Oujda, 2022)In this study, some important ADME parameters such as physicochemical properties, lipophilicity, water solubility, pharmacokinetics, medicinal chemistry and drug-likeness properties of ten triazole derivative compounds, ... -
Ternary transition metal complexes with an azo-imine Lligand and 2,2'-bipyridine: Characterization, computational calculations, and acetylcholinesterase inhibition activities
(Slovensko Kemijsko Drustvo, 2022)New mononuclear ternary transition metal complexes: [M(HL)(bipy)2]ClO4, (M: Mn(II) for 1, Ni(II) for 2), [M(HL) (bipy) (ClO4)], (M: Ni(II) for 3, Cu(II) for 4, Zn(II) for 5) with M(II), 2-[(hydroxyimino)methyl]-4-[-phenyldiazenyl] ... -
Urease and acetylcholinesterase enzyme inhibitor novel phthalonitrile azo compounds
(Scientific Publishers, 2022)Based on the relationship between Helicobacter pylori and Alzehimer's disease, new azo phthalonitrile compounds containing different amino pyridines have been synthesized. These compounds can inhibit both Urease and ... -
Synthesis and docking studies of novel benzimidazole derivatives containing thiophene and triazole rings as potential urease inhibitors
(Springer, 2022)Abstract: A new series of 5,6-dichloro-benzimidazoles containing thiophene ring derivatives of thiosemicarbazides and triazoles were designed, synthesized and characterized by spectral methods like as IR, 1H-NMR, 13C-NMR ... -
Some characteristics of new and innovative COX inhibitor derivatives: Potent hCA-I and hCA-II inhibitors supported by molecular docking studies
(John & Wiley Ltd., 2022)In this study, two novel metallophthalocyanines (ZnPc and CoPc) were synthesized using the corresponding metal salts 4-(4-(4-[4-chlorophenyl]-5-methylisoxazol-3-yl)phenoxy)-phthalonitrile (11), prepared from the reaction ... -
Synthesis of Benzimidazole derivatives containing Schiff base exhibiting antiurease activities
(Sivas Cumhuriyet Üniversitesi, 2021)In this study some novel Schiff bases derivatives of benzimidazole containing thiophene ring were designed and synthesized by using various aldehydes. Seven different aromatic aldehydes with various side groups were used ... -
The effect of usnea longissima extract on lung cancer cell line (A549)
(2021)Objective: Some lichens are known to demonstrate anticancer activity. However, to the best of our knowledge, no information is available about the activity of Usnea longissima against human lung cancer A549 cells. This ... -
Some azo compounds containing black tea processing waste catechins as antioxidant and urease enzyme inhibitory
(TUBİTAK Scientific & Technical Research Council Turkey, 2022)Although a lot of azo compounds containing some natural origin catechins had been synthesized and determined their dyeing properties for various textile products, the azo compounds containing black tea processing waste ... -
Peripheral or nonperipheral tetra-[4-(9H-carbazol-9-yl)phenoxy] substituted cobalt(II), manganese(III) phthalocyanines: Synthesis, acetylcholinesterase, butyrylcholinesterase, and α-glucosidase inhibitory effects and anticancer activities
(Wiley, 2020)In this work, peripheral or nonperipheral tetra-[4-(9H-carbazol-9-yl)phenoxy] substituted cobalt(II), manganese (III) phthalocyanines were synthesized for the first time. Their acetylcholinesterase from Electrophorus ... -
Synthesis of nonperipherally tetra-[5-(diethylamino)-2-formylphenoxy] substituted metallophthalocyanines and their electrochemistry
(TUBITAK, 2021)3-[5-(diethylamino)-2-formylphenoxy]phthalonitrile (n-TY-CN), metallophthalocyanines n-TY-Co, n-TY-Cu, and n-TY-Mn bearing [5-(diethylamino)-2-formylphenoxy] groups at nonperipheral positions were prepared for the first ... -
Novel fumarate derivatives synthesis and investigation of acetylcholinesterase inhibitor properties
(TUBİTAK Scientific & Technical Research Council Turkey, 2021)In this study, new fumarate compounds (I-IV) containing some natural phenols (eugenol, guaiacol, isoeugenol and vanillin) were synthesized and characterized. The single crystal X-ray diffraction technique was used to ... -
In silico inhibition potential of artemisinin derivatives against SARS-CoV-2 main protease
(TUBİTAK Scientific & Technical Research Council Turkey, 2021)The outbreak of COVID-19 caused by the SARS-CoV-2 virus has recently affected millions worldwide. The natural compounds obtained from medicinal plants have been proven to be the source of many treatments throughout history. ... -
Iron(III) complexes derived from azo-containing salicylaldoxime ligands: Synthesis, structures and biological evaluations
(TUBİTAK Scientific & Technical Research Council Turkey, 2021)Two novel mononuclear Fe(III) complexes derived from azo-containing salicylaldoxime ligands were synthesized and characterized by elemental analyses, spectroscopic data i.e. IR, 1H NMR, UV-Vis, electrospray ionization mass ... -
Α-glucosidase and α-amylase inhibition of some ethanolic propolis samples
(Bursa Uludag University, 2021)Propolis is a natural product, and it is of a great interest due to the possible uses of non-synthetic supplements in improving metabolic disorders. To support this claim, the current study was designed and presented. In ... -
Novel coumarin derivatives containing a triazole moiety: A study on synthesis, cytotoxicity, membrane dysfunction, apoptosis, cell cycle, and antiangiogenic effects
(Bentham Science Publications, 2022)Background: Coumarin is a functional compound with a pronounced wide range of biological activities and has recently been shown to have anticancer effects on various human cancer cells. Cisplatin is widely used in treating ... -
Sucrose-based activated carbon foams as an electrode active material for supercapacitors
(Springer, 2022)Activated carbon foams (ACFs) have been successfully prepared by foaming sucrose with Zn nitrate and further chemical activation with H3PO4. The effect of the foaming agent (Zn) concentration and the activation temperature ... -
Novel peripheral and non-peripheral oxobenzo[d]thiazol substituted cobalt phthalocyanines: Synthesis, electrochemistry, spectroelectrochemistry, electrocatalytic hydrogen production in alkaline medium
(Elsevier, 2022)In this study novel oxobenzo[d]thiazol substituted cobalt phthalocyanine complexes were synthesized and characterized by FT-IR, NMR, UV-vis spectroscopy, and mass spectrometry. The redox properties of peripheral and ... -
Elucidation of Bioactive compounds in flower extracts of Camellia sinensis by HPLC-DAD-MS/MS and their inhibitory effects on replicative bacterial DNA polymerases
(Elsevier, 2022)Camellia sinensis L. (C. sinensis) is an economically valuable crop whose leaves are used to produce tea. Tea flowers extracts (TFE) have been tested for their DNA polymerase inhibitory effect experimentally and in silico. ...
